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南开大学物理化学专业博士。现任首都医科大学教授,博士生导师。主要研究领域为材料药物化学,其主攻方向是抗肿瘤载药体系的设计合成。已在国外 J. Phys. Chem B., MedChemComm(封面文章)., Nanomedicine: Nanotechnology, Biology, and Medicine., Chem. Res. Toxicol. Nano Lett., J. Org. Chem., Chem-Eur. J.,发表文章。此外有5项专利授权。团队先后获得北京市人才专项、北京市教委科技面上项目、北京市中青年骨干教师、北京市科技新星、北京市青年拔尖人才培育计划、国家自然科学基金、国家科技重大专项课题/企业创新药物孵化基地建设、北京市创新团队、北京市自然基金等项目资助。
1.21103115,异喹啉生物碱与环糊精偶联物的超分子组装与抗血栓活性研究,李莉,国家自然科学基金,25万,2012.01-2014.12
2.2102013,环糊精-抗血栓药物偶联物的超分子组装及生物活性研究,李莉,北京市自然科学基金,11万,2010.01-2012.12
3.2172018,基于环糊精的多价态结合智能抗肿瘤药物载体的构筑,李莉,北京市自然科学基金,20万,2017.01-2019.12
4.2009A048,李莉,北京市科技新星,8万,2010.01-2012.12
发表文章:
1. Xueyuan Chen, Yi Zheng, Songlin Song, Ying Liu, Yi Wang, Yong Huang, Xiaoyi Zhang, Meng Zhang, Ming Zhao, Yuji Wang,* Li Li*.Design and Synthesis of Biotinylated Bivalent Carboline Derivatives as Potent Anti-tumor Agents. J. Org. Chem.. 2020,85:11618-11625.SCI
2. Fei Gao, Haiqing Liu, Li Li, Jianpeng Guo , Yuji Wang , Ming Zhao , Shiqi Peng.Design, synthesis, and testing of an isoquinoline-3- carboxylic –based novel anti-tumor lead. Bioorg. Med. Chem. Lett.. 2015,25:4434-4436.SCI
3. Li Li, Ming Zhao*, Wenhao Li, Yuji Wang, Zhuge Zhang, Ran An, Shiqi Peng*.Self-Complexation and Complexation Controlled Target Cancer Therapy. MedChemComm. 2012,3:2012, 1059-1061.SCI
4. Li Li, Ming Zhao*, Wenhao Li, Yuji Wang, Chunna Liu, Zhuge Zhang, Songchun Su, Shiqi Peng*.pH-Dependent nanostructure based on isoquinoline-cyclodextrin conjugate for thrombosis therapy. Nanomed-Techl.. 2012,8:2012, 8, 1216-1222.SCI
5. Li Li, Guohui Cui, Ming Zhao*, Yuji Wang, Hong Wang, Wei Li, Shiqi Peng*.Assembly of β-Cyclodextrin with 3S-Tetrahydro-β-carboline-3-carboxylic Acid and Self-Assembly of 6-(3’S-Carboline-3’-β-carboxylaminoethylamino)-6-deoxy-β-cyclodextrin: Approaches to Enhance Anti-Oxidation Stability and Anti-Thrombotic Potency. J. Phys. Chem. B. 2008,112:12139-12147.SCI
授权专利:
1. 李莉 赵明 彭师奇 马秋冉,七(6-(异喹啉-3-酰胺基)-6-脱氧)-β-环糊精及其制备方法和应用,授权号:ZL2014102552389
2.李莉,赵明,张海峰 全-6-(3’S-四氢异喹啉-3’-羧基氨基)-6-脱氧-β-环糊精 的制备及应用。授权号:ZL201210058813.7
3.李莉;赵明;王玉记;安然,四氢-β-咔啉-3-甲酰-二乙烯三胺-β-环糊精络铜,其制备,抗血栓作用和应用,授权号:ZL 201210181008.3
4.李莉、赵明、彭师奇、粟颂纯,β-环糊精修饰的四氢-β-咔啉羧酸衍生物及其制备方法, 授权号:ZL 201110164556.0
5. 李莉,赵明,李文昊,张朱舸,6-(1-甲基-β-咔啉-3-羧酸乙酰基)-6-脱氧-β-环糊精及其与阿霉素超分子包结配合物的制备和应用,授权号:ZL 201110237056.5
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